..., reversible, and high-affinity binding of compound 1 to human, mouse, and rat MT 2 melatonin receptors. cAMP, ERK1/2, and PathHunter β-arrestin recruitment assays revealed partial agonist activities. However, compound 1 induced a more intense internalization of human MT 2 melatonin receptor than melatonin...

... to persons or property resulting from any ideas, methods, instructions or products referred to in the content or advertisements. α 1 -Adrenoceptors Pithed rats Pertussis toxin G proteins Full agonist Partial agonist Imidazolines Phenethylamines Original Paper Pharmacology 1992;45:338-344...

...-adrenoceptors Calcium channel activator Intrinsic activity Full agonist Partial agonist Pharmacology 35: 272-278 (1987) Sensitivity of a-Adrenoceptor Agonists to the Calcium Channel Activator, Bay K 8644, in Canine Saphenous Vein Hanna Eskinder, Garrett J. Gross Department of Pharmacology and Toxicology...

.... Dihydroergotamine Dihydroergotoxin Noradrenaline Human femoral veins Human femoral arteries Antiadrenergic effect Partial agonist Pharmacology 24: 287-293 (1982) Dual Effect of Dihydroergotamine and Dihydroergotoxin in Isolated Human Femoral Veins and Arteries Erika Glusa, F. Markwardt Institute...

...Takahiro Horinouchi; Katsuo Koike (±)-Pindolol ([1-(1H-indol-4-yloxy)-3-[(1-methylethyl)- amino]-2-propanol)]) is a partial agonist at atypical β-adrenoceptors in the guinea pig gastric fundus. (±)-Pindolol induced concentration-dependent relaxation in this tissue. However, the relaxant responses...